Peptide News Digest

#Exatecan

2 stories

Clinical Trials · View digest

Avacta Details Phase 1 FOCUS-01 Trial of AVA6103, a FAP-Targeted Peptide-Drug Conjugate Carrying Exatecan, at AACR Pancreatic Cancer Conference

Avacta Group announced on Friday, September 25, 2026 that it would present the design of its Phase 1a FOCUS-01 trial and new preclinical data for AVA6103 (FAP-Exd) on September 26 at the AACR Conference on Pancreatic Cancer in San Diego. AVA6103 is a peptide-drug conjugate built on Avacta's pre|CISION platform, which is designed to be cleaved inside the tumor by fibroblast activation protein (FAP) so that the chemotherapy payload exatecan is released there, limiting exposure elsewhere in the body. The company said AVA6103 was well tolerated through the first three dose levels, up to a payload dose about 50% above the maximum tolerated dose of conventional exatecan, and that enrollment continues at dose level 4, including an every-two-weeks arm for pancreatic cancer. In mice implanted with human tumor tissue, Avacta reported durable complete and partial responses lasting weeks after dosing stopped; it released no efficacy data from patients.

Research · View digest

Avacta AVA6103 Peptide-Drug Conjugate Shows 3x Tumor Selectivity vs Enhertu in Preclinical Data

Avacta Therapeutics presented April 21 data at AACR 2026 showing its FAP-enabled peptide-drug conjugate AVA6103, which delivers exatecan via the pre|CISIONĀ® platform, achieved a Tumor Selectivity Index three times higher than marketed ADC Enhertu in preclinical models, with tumor Cmax more than one log higher. AVA6103 entered the Phase 1 FOCUS-01 trial (NCT07454642) in March 2026 with initial clinical readout expected later this year.